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Mechanism of Action of Pyridostigmine

mechanism of action of pyridostigmine

Introduction Pyridostigmine is a reversible acetylcholinesterase inhibitor of the quaternary ammonium carbamate class. It is primarily used to treat myasthenia gravis, reverse nondepolarizing neuromuscular blockade, and has a role in certain autonomic dysfunctions. Known for its peripheral action and minimal central nervous system penetration, pyridostigmine improves neuromuscular transmission by increasing acetylcholine availability at synapses. Mechanism … Read more

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